Name | PSNCBAM-1 |
---|---|
Supplier | Tocris Bioscience |
Catalog | 3353 |
Prices | $185.00, $755.00 |
Sizes | 10 mg, 50 mg |
Function Type | Modulator |
Cas Number | 877202-74-9 |
Chemical Name | N-(4-Chlorophenyl)-N'-[3-[6-(1-pyrrolidinyl)-2-pyridinyl]phenyl]urea |
Formula | C22H21ClN4O |
Molecular Weight | 392.88 |
Purity | >99 % |
Description | CB 1 receptor negative allosteric modulator (IC 50 values are 45 and 209 nM for the inhibition of CP 55,940 and WIN 55,212-2 respectively). Has no effect at the CB 2 receptor. Decreases food intake and body weight in rats. |
Supplier Page | Shop |
Horswill JG, Bali U, Shaaban S, Keily JF, Jeevaratnam P, Babbs AJ, Reynet C, Wong Kai In P. Br J Pharmacol. 2007 Nov;152(5):805-14. Epub 2007 Jun 25.
German N, Decker AM, Gilmour BP, Gay EA, Wiley JL, Thomas BF, Zhang Y. J Med Chem. 2014 Sep 25;57(18):7758-69.