L-R 4 W 2

Name L-R 4 W 2
Supplier Tocris Bioscience
Catalog 2144
Prices $225.00
Sizes 1 mg
Function Type Antagonist
Cas Number 206350-79-0
Formula C46H71N21O6
Molecular Weight 1014.2
Description Vanilloid TRPV1 (VR1) receptor antagonist peptide (IC 50 ~ 0.1 μ M); blocks Ca 2+ currents in dorsal root ganglion neurons. Analgesic in vivo .
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Product References

Arginine-rich peptides are blockers of VR-1 channels with analgesic activity. - Arginine-rich peptides are blockers of VR-1 channels with analgesic activity.

Planells-Cases R, Aracil A, Merino JM, Gallar J, Perez-Paya E, Belmonte C, Gonzalez-Ros JM, Ferrer-Montiel AV. FEBS Lett. 2000 Sep 15;481(2):131-6.

The arginine-rich hexapeptide R4W2 is a stereoselective antagonist at the - The arginine-rich hexapeptide R4W2 is a stereoselective antagonist at the

Himmel HM, Kiss T, Borvendeg SJ, Gillen C, Illes P. J Pharmacol Exp Ther. 2002 Jun;301(3):981-6.