Ritanserin

Name Ritanserin
Supplier Tocris Bioscience
Catalog 2443
Prices $69.00, $249.00
Sizes 10 mg, 50 mg
Function Type Antagonist
Cas Number 87051-43-2
Chemical Name 6-[2-[4-[Bis(4-fluorophenyl)methylene]-1-piperidinyl]ethyl]-7-methyl-5H-thiazolo[3,2-a]pyrimidin-5-one
Formula C27H25F2N3OS
Molecular Weight 477.57
Purity >99 %
Description Potent and long-acting 5-HT 2 receptor antagonist (K i = 0.39 nM). Anxiolytic in vivo .
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Product References

Pharmacology of potent and selective S2-serotonergic antagonists. - Pharmacology of potent and selective S2-serotonergic antagonists.

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Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and - Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and

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Syntheses and 5-HT2 antagonist activity of bicyclic 1,2,4-triazol-3(2H)-one and - Syntheses and 5-HT2 antagonist activity of bicyclic 1,2,4-triazol-3(2H)-one and

Watanabe Y, Usui H, Kobayashi S, Yoshiwara H, Shibano T, Tanaka T, Morishima Y, Yasuoka M, Kanao M. J Med Chem. 1992 Jan;35(1):189-94.