RWJ 52353

• Supplier: Tocris Bioscience
• Catalog: 4227
• Prices: $199.00
• Sizes: 10 mg
• Function Type: Agonist
• Cas Number: 245744-10-9
• Chemical Name: 5-(6,7-Dihydrobenzo[b]thien-4-yl-1H-imidazolehydrochloride
• Formula: C11H10N2S
• Molecular Weight: 202.28
• Purity: >98 %
• Description: Agonist of the α 2D adrenergic receptor (K i values are 1.5, 254, 443 and 621 nM for α 2D , α 2A , α 1 and α 2B adrenergic receptors respectively).

Product References

Alpha(2) adrenoceptor agonists as potential analgesic agents. 2. Discovery of - Alpha(2) adrenoceptor agonists as potential analgesic agents. 2. Discovery of

Ross TM, Jetter MC, McDonnell ME, Boyd RE, Connelly CD, Martinez RP, Lewis MA, Codd EE, Raffa RB, Reitz AB. J Med Chem. 2000 Apr 6;43(7):1423-6.

Inhibitory and facilitory actions of isocyanine derivatives at human and rat - Inhibitory and facilitory actions of isocyanine derivatives at human and rat

Amphoux A, Millan MJ, Cordi A, Bonisch H, Vialou V, Mannoury la Cour C, Dupuis DS, Giros B, Gautron S. Eur J Pharmacol. 2010 May 25;634(1-3):1-9.