Name | S 2101 |
---|---|
Supplier | Tocris Bioscience |
Catalog | 3911 |
Prices | $179.00, $745.00 |
Sizes | 10 mg, 50 mg |
Function Type | Inhibitor |
Cas Number | 1239262-36-2 |
Chemical Name | (1R,2S)-rel-2-[3,5-Difluoro-2-(phenylmethoxy)phenyl]cycloprpanaminehydrochloride |
Formula | C16H15F2NO.HCl |
Molecular Weight | 311.75 |
Purity | >98 % |
Description | LSD1 inhibitor (IC 50 = 990 nM; K i = 610 nM). Exhibits selectivity for LSD1 over MAO-B and MAO-A (K i values are 17 and 110 μ M, respectively). |
Supplier Page | Shop |
Beracochea D, Boucard A, Trocme-Thibierge C, Morain P. Psychopharmacology (Berl). 2008 Mar;196(4):555-64. Epub 2007 Nov 22.
Lagostena L, Trocme-Thibierge C, Morain P, Cherubini E. Neuropharmacology. 2008 Mar;54(4):676-85.
Marighetto A, Valerio S, Desmedt A, Philippin JN, Trocme-Thibierge C, Morain P. Psychopharmacology (Berl). 2008 Apr;197(3):499-508. doi: