SB 205607 dihydrobromide

• Supplier: Tocris Bioscience
• Catalog: 1512
• Prices: $249.00
• Sizes: 10 mg
• Function Type: Agonist
• Cas Number: 1217628-73-3
• Chemical Name: (R*,S*)-(±)-2-Methyl-4aa-(3-hydroxyphenyl)-1,2,3,4,4a,5,12,12aa-octahydroquinolino[2,3,3-g]isoquinolinedihydrobromide
• Formula: C23H24N2O.2HBr
• Molecular Weight: 506.28
• Purity: >97 %
• Description: The first described non-peptide δ 1 opioid receptor agonist with very high affinity and selectivity for the δ 1 subtype (K i values are 1.12, 2320 and 1790 nM at δ 1 , μ and κ receptors respectively).

Product References

Antinociceptive effects of the selective non-peptidic delta-opioid receptor - Antinociceptive effects of the selective non-peptidic delta-opioid receptor

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Properties of TAN-67, a nonpeptidic delta-opioid receptor agonist, at cloned - Properties of TAN-67, a nonpeptidic delta-opioid receptor agonist, at cloned

Knapp RJ, Landsman R, Waite S, Malatynska E, Varga E, Haq W, Hruby VJ, Roeske WR, Nagase H, Yamamura HI. Eur J Pharmacol. 1995 Oct 15;291(2):129-34.

The pharmacological profile of delta opioid receptor ligands, (+) and (-) TAN-67 - The pharmacological profile of delta opioid receptor ligands, (+) and (-) TAN-67

Nagase H, Yajima Y, Fujii H, Kawamura K, Narita M, Kamei J, Suzuki T. Life Sci. 2001 Apr 6;68(19-20):2227-31.