SC 26196

• Supplier: Tocris Bioscience
• Catalog: 1206
• Prices: $159.00, $665.00
• Sizes: 10 mg, 50 mg
• Function Type: Inhibitor
• Cas Number: 218136-59-5
• Chemical Name: α,α-Diphenyl-4-[(3-pyridinylmethylene)amino]-1-piperazinepentanenitrile
• Formula: C27H29N5
• Molecular Weight: 423.55
• Purity: >98 %
• Description: Selective Δ 6 desaturase inhibitor (IC 50 = 0.2 μ M in vitro ). Displays selectivity over Δ 5 and Δ 9 desaturases (IC 50 values are >200 μ M in vitro ). Exhibits anti-inflammatory properties in a mouse edema model. Eliminates CSCs from ovarian cancer cell lines and inhibits sphere formation in vitro .

Product References

Novel, selective delta6 or delta5 fatty acid desaturase inhibitors as - Novel, selective delta6 or delta5 fatty acid desaturase inhibitors as

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Selective inhibition of Delta-6 desaturase impedes intestinal tumorigenesis. - Selective inhibition of Delta-6 desaturase impedes intestinal tumorigenesis.

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A multiplexed cell assay in HepG2 cells for the identification of delta-5, - A multiplexed cell assay in HepG2 cells for the identification of delta-5,

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