| Name | SCH 442416 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 2299 |
| Prices | $95.00, $199.00, $825.00 |
| Sizes | 1 mg, 10 mg, 50 mg |
| Function Type | Antagonist |
| Cas Number | 316173-57-6 |
| Chemical Name | 2-(2-Furanyl)-7-[3-(4-methoxyphenyl)propyl]-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine |
| Formula | C20H19N7O2 |
| Molecular Weight | 389.42 |
| Purity | >99 % |
| Description | Selective adenosine A 2A receptor antagonist; binds to human and rat A 2A receptors with high affinity (K i values are 0.048 and 0.5 nM respectively). Displays > 23000-fold selectivity for hA 2A over hA 1 in vitro with minimal affinity for hA 2B and hA 3 receptors (IC 50 > 10 μ M). Blocks the cytoprotective effect of A 2A agonist CGS-21680 (Cat.No. 1063). |
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