SLIGKV-NH2

• Supplier: Tocris Bioscience
• Catalog: 1969
• Prices: $139.00
• Sizes: 5 mg
• Function Type: Agonist
• Cas Number: 190383-13-2
• Formula: C28H54N8O7
• Molecular Weight: 614.78
• Description: Protease-activated receptor 2 (PAR 2 ) agonist (K i = 9.64 μ M and IC 50 = 10.4 μ M). Corresponds to the tethered ligand exposed by trypsin cleavage of PAR-2. Control peptide VKGILS-NH 2 also available (Cat. No. 3392).

Product References

Molecular cloning, expression and potential functions of the human - Molecular cloning, expression and potential functions of the human

Bohm SK, Kong W, Bromme D, Smeekens SP, Anderson DC, Connolly A, Kahn M, Nelken NA, Coughlin SR, Payan DG, Bunnett NW. Biochem J. 1996 Mar 15;314 ( Pt 3):1009-16.

International Union of Pharmacology. XXVIII. Proteinase-activated receptors. - International Union of Pharmacology. XXVIII. Proteinase-activated receptors.

Hollenberg MD, Compton SJ. Pharmacol Rev. 2002 Jun;54(2):203-17.

Binding of a highly potent protease-activated receptor-2 (PAR2) activating - Binding of a highly potent protease-activated receptor-2 (PAR2) activating

Kanke T, Ishiwata H, Kabeya M, Saka M, Doi T, Hattori Y, Kawabata A, Plevin R. Br J Pharmacol. 2005 May;145(2):255-63.