Name | SNC 162 |
---|---|
Supplier | Tocris Bioscience |
Catalog | 3347 |
Prices | $225.00, $925.00 |
Sizes | 10 mg, 50 mg |
Function Type | Agonist |
Cas Number | 178803-51-5 |
Chemical Name | 4-[(S)-[(2S,5R)-2,5-Dimethyl-4-(2-propenyl)-1-piperazinyl]phenylmethyl]-N,N-diethylbenzamide |
Formula | C27H37N3O |
Molecular Weight | 419.61 |
Purity | >99 % |
Description | Potent and selective non-peptide δ -opioid receptor agonist (K i = 0.63 nM). Displays > 8000-fold selectivity over μ -opioid receptors and is centrally active following systemic administration in vivo . |
Supplier Page | Shop |
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Calderon SN, Rice KC, Rothman RB, Porreca F, Flippen-Anderson JL, Kayakiri H, Xu H, Becketts K, Smith LE, Bilsky EJ, Davis P, Horvath R. J Med Chem. 1997 Feb 28;40(5):695-704.
Negus SS, Gatch MB, Mello NK, Zhang X, Rice K. J Pharmacol Exp Ther. 1998 Jul;286(1):362-75.