| Name | TC OT 39 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 5087 |
| Prices | $245.00 |
| Sizes | 10 mg |
| Function Type | Agonist |
| Cas Number | 479232-57-0 |
| Chemical Name | (2S)-N-[[4-[(4,10-Dihydro-1-methylpyrazolo[3,4-b][1,5]benzodiazepin-5(1H)-yl)carbonyl]-2-methylphenyl]methyl]-2-[(hexahydro-4-methyl-1H-1,4-diazepin-1-yl)thioxomethyl]-1-pyrrolidinecarboxamide |
| Formula | C32H40N8O2S |
| Molecular Weight | 600.78 |
| Purity | >97 % |
| Description | Potent non-peptide oxytocin receptor partial agonist (EC 50 values are 33 nM and 850 nM for the oxytocin receptor and V 2 vasopressin receptor respectively). Also a V 1a vasopressin receptor antagonist (K i = 330 nM). Active in vivo in a rat model of uterine response. |
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