| Name | TC-G 1008 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 4747 |
| Prices | $195.00, $805.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Agonist |
| Cas Number | 1621175-65-2 |
| Chemical Name | N-[3-Chloro-4-[[[2-(methylamino)-6-(2-pyridinyl)-4-pyrimidinyl]amino]methyl]phenyl]methanesulfonamide |
| Formula | C18H19ClN6O2S |
| Molecular Weight | 418.9 |
| Purity | >98 % |
| Description | Potent and selective GPR39 agonist (EC 50 values are 0.4 and 0.8 nM for rat and human receptors respectively). Selective over a panel of kinases (IC 50 s > 10 μ M) and displays minimal binding affinity for ghrelin and neurotensin-1 receptors (IC 50 s > 30 μ M). Increases GLP-1 levels in vitro and in vivo . Orally bioavailable. |
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