Name | TC-N 1752 |
---|---|
Supplier | Tocris Bioscience |
Catalog | 4365 |
Prices | $225.00, $925.00 |
Sizes | 10 mg, 50 mg |
Function Type | Blocker |
Cas Number | 1211866-85-1 |
Chemical Name | N-[2-Methyl-3-[[4-[4-[[4-(trifluoromethoxy)phenyl]methoxy]-1-piperidinyl]-1,3,5-triazin-2-yl]amino]phenyl]acetamide |
Formula | C25H27F3N6O3 |
Molecular Weight | 516.52 |
Purity | >99 % |
Description | Selective blocker of human Na V 1.7 channels (IC 50 values are 0.17, 0.3, 0.4 and 1.1 μ M at hNa V 1.7, hNa V 1.3, hNa V 1.4 and hNa V 1.5 respectively). Also inhibits tetrodotoxin-sensitive sodium channels. Displays analgesic efficacy in the formalin pain model. |
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