Name | TCS 1102 |
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Supplier | Tocris Bioscience |
Catalog | 1225 |
Prices | $159.00, $665.00 |
Sizes | 10 mg, 50 mg |
Function Type | Antagonist |
Cas Number | 916141-36-1 |
Chemical Name | N-[1,1'-Biphenyl]-2-yl-1-[2-[(1-methyl-1H-benzimidazol-2-yl)thio]acetyl-2-pyrrolidinedicarboxamide |
Formula | C27H26N4O2S |
Molecular Weight | 470.59 |
Purity | >98 % |
Description | Potent, dual orexin receptor antagonist (K i values are 0.2 and 3 nM for OX 2 and OX 1 receptors respectively). Inhibits ADL-orexin B-mediated locomotion following i.p. administration in vivo . Brain penetrant. |
Supplier Page | Shop |