| Name | TCS ERK 11e |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 5286 |
| Prices | $255.00 |
| Sizes | 10 mg |
| Function Type | Inhibitor |
| Cas Number | 896720-20-0 |
| Chemical Name | 4-[2-[(2-Chloro-4-fluorophenyl)amino]-5-methyl-4-pyrimidinyl]-N-[(1S)-1-(3-chlorophenyl)-2-hydroxyethyl]-1H-pyrrole-2-carboxamide |
| Formula | C24H20Cl2FN5O2 |
| Molecular Weight | 500.35 |
| Purity | >98 % |
| Description | Potent and selective extracellular signal-related kinase 2 (ERK2) inhibitor (K i values are <2, 395, 540 and 852 nM for ERK2, GSK-3, Aurora Kinase A and Cdk2 respectively). Potently blocks proliferation of HT29 cells (IC 50 = 48 nM). Orally bioavailable. |
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