| Name | TCS PIM-1 4a |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 2979 |
| Prices | $99.00, $419.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Inhibitor |
| Cas Number | 438190-29-5 |
| Chemical Name | (5Z)-5-[[3-(Trifluoromethyl)phenyl]methylene]-2,4-thiazolidinedione |
| Formula | C11H6F3NO2S |
| Molecular Weight | 273.23 |
| Purity | >98 % |
| Description | Selective, ATP-competitive Pim kinase inhibitor (IC 50 values are 24 and 100 nM for Pim-1 and Pim-2 respectively). Displays selectivity over a panel of ~50 other kinases tested. Exhibits cytotoxicity in PC3 prostate carcinoma cells in vitro (IC 50 = 17 μ M). |
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