Telenzepine dihydrochloride

• Supplier: Tocris Bioscience
• Catalog: 3664
• Prices: $69.00, $255.00
• Sizes: 10 mg, 50 mg
• Function Type: Antagonist
• Cas Number: 147416-96-4
• Chemical Name: 4,9-Dihydro-3-methyl-4-[(4-methyl-1-piperazinyl)acetyl]-10H-thieno[3,4-b][1,5]benzodiazepin-10-onedihydrochloride
• Formula: C19H22N4O2S.2HCl
• Molecular Weight: 443.39
• Description: Selective high affinity muscarinic M 1 receptor antagonist (K i = 0.94 nM). Inhibits gastric acid secretion.

Product References

Pharmacological evidence for selective inhibition of gastric acid secretion by - Pharmacological evidence for selective inhibition of gastric acid secretion by

Eltze M, Gonne S, Riedel R, Schlotke B, Schudt C, Simon WA. Eur J Pharmacol. 1985 Jun 7;112(2):211-24.

Interaction of telenzepine with muscarinic receptors in mammalian sympathetic - Interaction of telenzepine with muscarinic receptors in mammalian sympathetic

Galvan M, Boer R, Schudt C. Eur J Pharmacol. 1989 Aug 11;167(1):1-10.

Neuropharmacology of the muscarinic antagonist telenzepine in myenteric ganglia - Neuropharmacology of the muscarinic antagonist telenzepine in myenteric ganglia

Christofi FL, Palmer JM, Wood JD. Eur J Pharmacol. 1991 Apr 3;195(3):333-9.