TGX 221

• Supplier: Tocris Bioscience
• Catalog: 5425
• Prices: $255.00, $1,045.00
• Sizes: 10 mg, 50 mg
• Function Type: Inhibitor
• Cas Number: 663619-89-4
• Chemical Name: 7-Methyl-2-(4-morpholinyl)-9-[1-(phenylamino)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one
• Formula: C21H24N4O2
• Molecular Weight: 364.44
• Purity: >98 %
• Description: Potent and selective PI 3-kinase β inhibitor (IC 50 values are 0.007, 0.1, 3.5 and 5 μ M for the β , δ , γ and α isoforms, respectively). Shows >1,000-fold selectively for PI 3-kinase β over a range of other kinases. Inhibits thrombus formation in animal models.

Product References

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