Urapidil hydrochloride

Name Urapidil hydrochloride
Supplier Tocris Bioscience
Catalog 5296
Prices $139.00
Sizes 100 mg
Function Type Antagonist
Cas Number 64887-14-5
Chemical Name 6-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]amino]-1,3-dimethyl-2,4(1H,3H)-pyrimidinedionehydrochloride
Formula C20H29N5O3.HCl
Molecular Weight 423.94
Purity >99 %
Description α 1 -adrenoceptor antagonist and 5-HT 1A receptor agonist (pIC 50 values are 6.13 and 6.4 respectively). Clinically used hypotensive agent.
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Product References

Urapidil and some analogues with hypotensive properties show high affinities for - Urapidil and some analogues with hypotensive properties show high affinities for

Gross G, Hanft G, Kolassa N. Naunyn Schmiedebergs Arch Pharmacol. 1987 Dec;336(6):597-601.

Involvement of brain 5-HT1A receptors in the hypotensive response to urapidil. - Involvement of brain 5-HT1A receptors in the hypotensive response to urapidil.

Kolassa N, Beller KD, Sanders KH. Am J Cardiol. 1989 Aug 15;64(7):7D-10D.

Pharmacologic profile of urapidil. - Pharmacologic profile of urapidil.

van Zwieten PA. Am J Cardiol. 1989 Aug 15;64(7):1D-6D.