[Orn 5 ]-URP

• Supplier: Tocris Bioscience
• Catalog: 1642
• Prices: $189.00
• Sizes: 1 mg
• Function Type: Antagonist
• Cas Number: 782485-03-4
• Formula: C48H62N10O10S2
• Molecular Weight: 1003.2
• Description: Urotensin-II (UT) receptor pure antagonist (pEC 50 = 7.24). Displays no agonist activity unlike other U-II/URP analogs. Inhibits the action of U-II in the rat aorta ring assay.

Product References

Structure-activity relationships and structural conformation of a novel urotensin - Structure-activity relationships and structural conformation of a novel urotensin

Chatenet D, Dubessy C, Leprince J, Boularan C, Carlier L, Segalas-Milazzo I, Guilhaudis L, Oulyadi H, Davoust D, Scalbert E, Pfeiffer B, Renard P, Tonon MC, Lihrmann I, Pacaud P, Vaudry H. Peptides. 2004 Oct;25(10):1819-30.

[Orn5]URP acts as a pure antagonist of urotensinergic receptors in rat cortical - [Orn5]URP acts as a pure antagonist of urotensinergic receptors in rat cortical

Diallo M, Jarry M, Desrues L, Castel H, Chatenet D, Leprince J, Vaudry H, Tonon MC, Gandolfo P. Peptides. 2008 May;29(5):813-9. Epub 2007 Nov 6.