Name | VU 0255035 |
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Supplier | Tocris Bioscience |
Catalog | 3888 |
Prices | $175.00, $709.00 |
Sizes | 10 mg, 50 mg |
Function Type | Antagonist |
Cas Number | 1135243-19-4 |
Chemical Name | N-[3-Oxo-3-[4-(4-pyridinyl)-1-piperazinyl]propyl]-2,1,3-benzothiadiazole-4-sulfonamide |
Formula | C18H20N6O3S2 |
Molecular Weight | 432.52 |
Purity | >99 % |
Description | Highly selective muscarinic M 1 antagonist (K i = 14.87 nM). Targets the M 1 orthosteric site with greater than 75-fold selectivity over the other receptor subtypes. Reduces pilocarpine-induced seizures in mice. Brain penetrant. |
Supplier Page | Shop |