Zinterol hydrochloride

• Supplier: Tocris Bioscience
• Catalog: 0746
• Prices: $169.00, $705.00
• Sizes: 10 mg, 50 mg
• Function Type: Agonist
• Cas Number: 37000-20-7
• Chemical Name: N-[5-[2-[(1,1-Dimethyl-2-phenylethyl)amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulphonamidehydrochloride
• Formula: C19H26N2O4S
• Molecular Weight: 414.95
• Purity: >98 %
• Description: Potent and selective β 2 -adrenoceptor agonist (pK B values are 8.3 and < 5.7 for β 2 and β 1 receptors respectively, as measured in human artery).

Product References

Beta-2 adrenergic activation of L-type Ca++ current in cardiac myocytes. - Beta-2 adrenergic activation of L-type Ca++ current in cardiac myocytes.

Skeberdis VA, Jurevicius J, Fischmeister aR. J Pharmacol Exp Ther. 1997 Nov;283(2):452-61.

Four beta-adrenoceptor subtypes in the mammalian heart. - Four beta-adrenoceptor subtypes in the mammalian heart.

Kaumann AJ. Trends Pharmacol Sci. 1997 Mar;18(3):70-6.

Agonist effects of zinterol at the mouse and human beta(3)-adrenoceptor. - Agonist effects of zinterol at the mouse and human beta(3)-adrenoceptor.

Hutchinson DS, Chernogubova E, Sato M, Summers RJ, Bengtsson T. Naunyn Schmiedebergs Arch Pharmacol. 2006 May;373(2):158-68. Epub 2006 Apr 7.