RG 102240

• Supplier: Tocris Bioscience
• Catalog: 5677
• Prices: $139.00, $585.00
• Sizes: 10 mg, 50 mg
• Cas Number: 162326-49-0
• Chemical Name: 2-Ethyl-3-methoxybenzoicacid2-(3,5-dimethylbenzoyl)-2-(1,1-dimethylethyl)hydrazide
• Formula: C23H30N2O3
• Molecular Weight: 382.5
• Purity: >98 %
• Description: Gene switch ligand. Transcription inducer for use in induceable gene expression systems. Does not cause significant changes in endogenous gene expression in HEK cells.

Product References

Epigenetic reactivation of tumor suppressor genes by a novel small-molecule - Epigenetic reactivation of tumor suppressor genes by a novel small-molecule

Brueckner B, Garcia Boy R, Siedlecki P, Musch T, Kliem HC, Zielenkiewicz P, Suhai S, Wiessler M, Lyko F. Cancer Res. 2005 Jul 15;65(14):6305-11.

Synthesis and in vitro evaluation of biotinylated RG108: a high affinity compound - Synthesis and in vitro evaluation of biotinylated RG108: a high affinity compound

Schirrmacher E, Beck C, Brueckner B, Schmitges F, Siedlecki P, Bartenstein P, Lyko F, Schirrmacher R. Bioconjug Chem. 2006 Mar-Apr;17(2):261-6.

Functional diversity of DNA methyltransferase inhibitors in human cancer cell - Functional diversity of DNA methyltransferase inhibitors in human cancer cell

Stresemann C, Brueckner B, Musch T, Stopper H, Lyko F. Cancer Res. 2006 Mar 1;66(5):2794-800.