| Name | SR 8278 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 5626 |
| Prices | $175.00, $709.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Antagonist |
| Cas Number | 1254944-66-5 |
| Chemical Name | 1,2,3,4-Tetrahydro-2-[[5-(methylthio)-2-thienyl]carbonyl]-3-isoquinolinecarboxylicacidethylester |
| Formula | C18H19NO3S2 |
| Molecular Weight | 361.48 |
| Purity | >99 % |
| Description | Rev-Erb α antagonist; inhibits Rev-Erb α transcriptional repression (EC 50 = 0.47 μ M). Blocks activity of Rev-Erb α agonist GSK 4112 (Cat. No. 3663) in HEK293 cells. Increases expression of glucose-regulating genes, G6Pase and PEPCK in HepG2 cells. |
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