Name | VU 0409551 |
---|---|
Supplier | Tocris Bioscience |
Catalog | 5322 |
Prices | $179.00, $745.00 |
Sizes | 10 mg, 50 mg |
Function Type | Modulator |
Cas Number | 1363281-27-9 |
Chemical Name | [6,7-Dihydro-2-(phenoxymethyl)oxazolo[5,4-c]pyridin-5(4H)-yl](fluorophenyl)methanone |
Formula | C20H17FN2O3 |
Molecular Weight | 352.36 |
Purity | >98 % |
Description | Selective mGlu 5 positive allosteric modulator (EC 50 = 260 nM). Selective for mGlu 5 over other mGluR subtypes, as well as 66 other receptors and ion channels. Selectively potentiates mGlu 5 signaling via G α q . Exhibits wake-promoting, antipsychotic-like and cognition-enhancing effects in animal models. Brain penetrant and orally available. |
Supplier Page | Shop |