BIBN 4096

Name BIBN 4096
Supplier Tocris Bioscience
Catalog 5590
Prices $289.00
Sizes 10 mg
Function Type Antagonist
Cas Number 204697-65-4
Chemical Name 1-[3,5-Dibromo-N-[[4-(1,4-dihydro-2-oxo-3(2H)-quinazolinyl)-1-piperidinyl]carbonyl]-D-tyrosyl-L-lysyl]-4-(4-pyridinyl)-piperazine
Formula C38H47Br2N9O5
Molecular Weight 869.65
Purity >95 %
Description Potent and selective CGRP receptor antagonist (IC 50 values are 0.03 and 6.4 nM for human and rat CGRP receptors respectively). Displays high affinity for human CGRP receptors (K i = 14.4 pM); exhibits no significant affinity for 75 other receptors.
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