| Name | CGH 2466 dihydrochloride |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 5946 |
| Prices | $139.00, $585.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Antagonist |
| Cas Number | 1177618-54-0 |
| Chemical Name | 4-(3,4-Dichlorophenyl)-5-(4-pyridinyl)-2-thiazolaminedihydrochloride |
| Formula | C14H9N3SCl2.2HCl |
| Molecular Weight | 395.13 |
| Purity | >99 % |
| Description | Adenosine A 1 , A 2B and A 3 receptor antagonist (IC 50 values are 19, 21, and 80 nM respectively). Also inhibits p38 MAPK (IC 50 = 187 - 400 nM) and phosphodiesterase type 4D (IC 50 = 22 nM). Displays potent anti-inflammatory effects in vitro and in vivo . Potentially useful for asthma and chronic obstructive pulmonary disease (COPD) research. |
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