SR 9243

• Supplier: Tocris Bioscience
• Catalog: 5854
• Prices: $149.00, $629.00
• Sizes: 10 mg, 50 mg
• Function Type: Agonist
• Cas Number: 1613028-81-1
• Chemical Name: N-[2-(3-Bromophenyl)ethyl]-2,4,6-trimethyl-N-[[3'-(methylsulfonyl)[1,1'-biphenyl]-4-yl]methyl]benzenesulfonamide
• Formula: C31H32BrNO4S2
• Molecular Weight: 626.62
• Purity: >98 %
• Description: Selective LXR inverse agonist. Exhibits no significant activity at other nuclear receptors at maximally effective concentration. Inhibits the Warburg effect and lipogenesis by down-regulation of LXR-mediated gene expression. Selectively reduces cell viability and induces apoptosis in cancer cell lines in vitro . Suppresses hepatic steatosis and inhibits growth of tumor xenografts in mice.