| Name | AR-C155858 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 5720 |
| Prices | $175.00 |
| Sizes | 1 mg |
| Function Type | Inhibitor |
| Cas Number | 496791-37-8 |
| Chemical Name | 6-[(3,5-Dimethyl-1H-pyrazol-4-yl)methyl]-5-[[(4S)-4-hydroxy-2-isoxazolidinyl]carbonyl]-3-methyl-1-(2-methylpropyl)thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione |
| Formula | C21H27N5O5S |
| Molecular Weight | 461.53 |
| Purity | >98 % |
| Description | Inhibitor of the monocarboxylate transporters (MCTs) MCT1 and MCT2 (K i values are 2.3 and <10 nM respectively). Exhibits no activity at MCT4. Blocks proliferation of Raji lymphoma cells in vitro . Inhibits glycolysis and glutathione synthesis in cancer cells. |
| Supplier Page | Shop |