GSK 5959

• Supplier: Tocris Bioscience
• Catalog: 5777
• Prices: $209.00, $879.00
• Sizes: 10 mg, 50 mg
• Function Type: Inhibitor
• Cas Number: 901245-65-6
• Chemical Name: N-[2,3-Dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxybenzamide
• Formula: C22H26N4O3
• Molecular Weight: 394.47
• Purity: >99 %
• Description: Potent and selective BRPF1 bromodomain inhibitor (IC 50 = 80 nM). Exhibits >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Inhibits BRPF1 interaction with histone H3.3. Cell permeable.