Lu AA 47070

• Supplier: Tocris Bioscience
• Catalog: 5835
• Prices: $199.00, $825.00
• Sizes: 10 mg, 50 mg
• Function Type: Antagonist
• Cas Number: 913842-25-8
• Chemical Name: 4-[(3,3-Dimethyl-1-oxobutyl)amino]-3,5-difluoro-N-[3-[(phosphonooxy)methyl]-2(3H)-thiazolylidene]benzamide
• Formula: C17H20F2N3O6PS
• Molecular Weight: 463.39
• Purity: >98 %
• Description: Prodrug of a potent and selective adenosine A 2A receptor antagonist (K i values are 5.9, 260, 410 and <10,000 nM for A 2A , A 2B , A 1 and A 3 receptors respectively. Reverses parkinsonian motor impairment and motivational effects produced by dopamine D 2 receptor blockade in rats. Orally bioavailable.