Name | LGK974 |
---|---|
Supplier | BioGems |
Catalog | 1241454 |
Prices | $65.00, $180.00 |
Sizes | 1 mg, 5 mg |
Function Type | Inhibitor |
Cas Number | 1243244-14-5 |
Chemical Name | 2-[5-methyl-6-(2-methylpyridin-4-yl)pyridin-3-yl]-N-(5-pyrazin-2-ylpyridin-2-yl)acetamide |
Formula | C23H20N6O |
Molecular Weight | 396.4 |
Purity | ≥98% |
Description | LGK974 is a highly potent inhibitor of Porcupine (PORCN), a Wnt-specific acyltransferase. LGK974 is orally bioavailable and inhibits WNT signaling in vitro and in vivo. It is reported to exhibit anti-tumor properties without increasing cytotoxicity. |
Supplier Page | Shop |