Gene Symbol | HTR2C |
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Entrez Gene | 3358 |
Alt Symbol | 5-HT1C, 5-HT2C, 5-HTR2C, 5HTR2C, HTR1C |
Species | Human |
Gene Type | protein-coding |
Description | 5-hydroxytryptamine (serotonin) receptor 2C, G protein-coupled |
Other Description | 5-hydroxytryptamine receptor 1C|5-hydroxytryptamine receptor 2C|serotonin 5-HT-1C receptor|serotonin 5-HT-2C receptor |
Swissprots | Q9NP28 Q5VUF8 P28335 B1AMW4 |
Accessions | AAC71658 ACE96318 ACE96323 ACE96328 CAB59978 EAX02623 EAX02624 P28335 AF208053 AAF35842 AF498983 AAM21130 AK295753 BAG58583 AK308766 AY114104 AAM78371 BC028688 BC095543 AAH95543 BX648587 FJ200493 ACO54890 M81778 AAA60317 U49516 AAB40898 NM_000868 NP_000859 NM_001256760 NP_001243689 NM_001256761 NP_001243690 |
Function | G-protein coupled receptor for 5-hydroxytryptamine (serotonin). Also functions as a receptor for various drugs and psychoactive substances, including ergot alkaloid derivatives, 1- 2,5,-dimethoxy-4-iodophenyl-2-aminopropane (DOI) and lysergic acid diethylamide (LSD). Ligand binding causes a conformation change that triggers signaling via guanine nucleotide-binding proteins (G proteins) and modulates the activity of down-stream effectors. Beta-arrestin family members inhibit signaling via G proteins and mediate activation of alternative signaling pathways. Signaling activates a phosphatidylinositol-calcium second messenger system that modulates the activity of phosphatidylinositol 3-kinase and down-stream signaling cascades and promotes the release of Ca(2+) ions from intracellular stores. Regulates neuronal activity via the activation of short transient receptor potential calcium channels in the brain, and thereby modulates the activation of pro-opiomelacortin neurons and the release o |
Subcellular Location | Cell membrane {ECO:0000269|PubMed:12970106, ECO:0000269|PubMed:18703043, ECO:0000269|PubMed:19057895, ECO:0000269|PubMed:7895773}; Multi-pass membrane protein {ECO:0000269|PubMed:12970106, ECO:0000269|PubMed:18703043, ECO:0000269|PubMed:19057895, ECO:0000269|PubMed:7895773}. |
Tissue Specificity | Detected in brain. {ECO:0000269|PubMed:8812491}. |
Top Pathways | Gap junction, Calcium signaling pathway, Inflammatory mediator regulation of TRP channels, Neuroactive ligand-receptor interaction |
SR-2C CRISPR/Cas9 KO Plasmid (h) - sc-400886 from Santa Cruz Biotechnology
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SR-2C HDR Plasmid (h) - sc-400886-HDR from Santa Cruz Biotechnology
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SR-2C Double Nickase Plasmid (h) - sc-400886-NIC from Santa Cruz Biotechnology
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SR-2C Double Nickase Plasmid (h2) - sc-400886-NIC-2 from Santa Cruz Biotechnology
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SR-2C CRISPR Activation Plasmid (h) - sc-400886-ACT from Santa Cruz Biotechnology
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SR-2C CRISPR Activation Plasmid (h2) - sc-400886-ACT-2 from Santa Cruz Biotechnology
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SR-2C Lentiviral Activation Particles (h) - sc-400886-LAC from Santa Cruz Biotechnology
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SR-2C Lentiviral Activation Particles (h2) - sc-400886-LAC-2 from Santa Cruz Biotechnology
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SR-2C siRNA (h) - sc-42235 from Santa Cruz Biotechnology
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SR-2C shRNA Plasmid (h) - sc-42235-SH from Santa Cruz Biotechnology
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SR-2C shRNA (h) Lentiviral Particles - sc-42235-V from Santa Cruz Biotechnology
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MISSION® esiRNA - EHU120291 from Sigma-Aldrich
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CompoZr® Knockout ZFN Kit - CKOZFN1830 from Sigma-Aldrich
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CompoZr® Knockout ZFN Kit, ZFN plasmid only - CKOZFND1830 from Sigma-Aldrich
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MISSION® 3′UTR Lenti GoClone™ - HUTR11673 from Sigma-Aldrich
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HTR2C siRNA (Human) - CRH2288 from Cohesion Biosciences
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5-HT2C RNAi - H00003358-R02 from Novus Biologicals
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HTR2C - MBS8224517 from MyBioSource
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SR-2C CRISPR/Cas9 KO Plasmid (h2) - sc-400886-KO-2 from Santa Cruz Biotechnology
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SR-2C HDR Plasmid (h2) - sc-400886-HDR-2 from Santa Cruz Biotechnology
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shRNA set against Human HTR2C (NM_000868.2) - SHH315937 from Creative biogene
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shRNA set against Human HTR2C(NM_000868.2) - SHH135749 from Creative biogene
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Human HTR2C siRNA - orb262790 from Biorbyt
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HTR2C shRNA Plasmid (Human) - CHH2288 from Cohesion Biosciences
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HTR2C miRNA 3'UTR clone - MiUTR1H-04754 from Creative biogene
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