Gene Symbol | OPRK1 |
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Entrez Gene | 4986 |
Alt Symbol | K-OR-1, KOR, KOR-1, OPRK |
Species | Human |
Gene Type | protein-coding |
Description | opioid receptor, kappa 1 |
Other Description | Opiate receptor, kappa-1|kappa opioid receptor|kappa-type opioid receptor |
Swissprots | E5RHC9 P41145 Q499G4 |
Accessions | AAA56758 EAW86723 P41145 AF498922 AAM21070 AK023198 AK310233 AK310407 AK313058 BAG35888 AY168006 AAN87342 AY466378 AAR36879 BC099912 AAH99912 BF061371 EF057067 L36130 AAA63646 L37362 AAA63906 U11053 AAA20985 U17298 AAC50158 NM_000912 NP_000903 NM_001282904 NP_001269833 |
Function | G-protein coupled opioid receptor that functions as receptor for endogenous alpha-neoendorphins and dynorphins, but has low affinity for beta-endorphins. Also functions as receptor for various synthetic opioids and for the psychoactive diterpene salvinorin A. Ligand binding causes a conformation change that triggers signaling via guanine nucleotide-binding proteins (G proteins) and modulates the activity of down-stream effectors, such as adenylate cyclase. Signaling leads to the inhibition of adenylate cyclase activity. Inhibits neurotransmitter release by reducing calcium ion currents and increasing potassium ion conductance. Plays a role in the perception of pain. Plays a role in mediating reduced physical activity upon treatment with synthetic opioids. Plays a role in the regulation of salivation in response to synthetic opioids. May play a role in arousal and regulation of autonomic and neuroendocrine functions. {ECO:0000269|PubMed:12004055, ECO:0000269|PubMed:22437504, ECO:0000269 |
Subcellular Location | Cell membrane {ECO:0000269|PubMed:12004055, ECO:0000269|PubMed:22437504, ECO:0000269|PubMed:7624359, ECO:0000269|PubMed:8060324}; Multi-pass membrane protein {ECO:0000269|PubMed:12004055, ECO:0000269|PubMed:22437504, ECO:0000269|PubMed:7624359, ECO:0000269|PubMed:8060324}. |
Tissue Specificity | Detected in brain and placenta. {ECO:0000269|PubMed:7624359, ECO:0000269|PubMed:8060324}. |
Top Pathways | Neuroactive ligand-receptor interaction |
KOR-1 (D-8) - sc-374479 from Santa Cruz Biotechnology
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KOR-1 (C-20) - sc-7493 from Santa Cruz Biotechnology
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KOR-1 (H-70) - sc-9112 from Santa Cruz Biotechnology
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KOR-1 (N-19) - sc-7494 from Santa Cruz Biotechnology
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Anti-Kappa Opioid Receptor antibody - ab113533 from Abcam
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Anti-Kappa Opioid Receptor antibody - ab137264 from Abcam
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Anti-Kappa Opioid Receptor antibody - ab109979 from Abcam
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Anti-Kappa Opioid Receptor antibody - C-terminal - ab179873 from Abcam
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Anti-Kappa Opioid Receptor antibody - N-terminal - ab194371 from Abcam
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Anti-OPRK1 / Kappa Opioid Receptor Antibody (aa366-380) IHC-plus⢠- LS-B6883 from LifeSpan Bioscience
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Anti-OPRK1 / Kappa Opioid Receptor Antibody (C-Terminus) - LS-C37882 from LifeSpan Bioscience
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Anti-OPRK1 / Kappa Opioid Receptor Antibody (C-Terminus) - LS-C37883 from LifeSpan Bioscience
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Anti-OPRK1 / Kappa Opioid Receptor Antibody (Internal, Azide-free) - LS-C37885 from LifeSpan Bioscience
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Anti-OPRK1 / Kappa Opioid Receptor Antibody (C-Terminus) - LS-C37884 from LifeSpan Bioscience
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Anti-OPRK1 / Kappa Opioid Receptor Antibody (Internal) - LS-C37886 from LifeSpan Bioscience
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Anti-OPRK1 / Kappa Opioid Receptor Antibody - LS-C37887 from LifeSpan Bioscience
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Anti-OPRK1 / Kappa Opioid Receptor Antibody (aa181-209, AP) - LS-C264999 from LifeSpan Bioscience
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Anti-OPRK1 / Kappa Opioid Receptor Antibody (N-Terminus) - LS-C102843 from LifeSpan Bioscience
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Anti-OPRK1 / Kappa Opioid Receptor Antibody (aa331-380) - LS-C199174 from LifeSpan Bioscience
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Anti-OPRK1 / Kappa Opioid Receptor Antibody (aa181-209, APC) - LS-C265000 from LifeSpan Bioscience
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Anti-OPRK1 / Kappa Opioid Receptor Antibody (aa312-361) - LS-C200300 from LifeSpan Bioscience
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Anti-OPRK1 / Kappa Opioid Receptor Antibody (aa181-209, Biotin) - LS-C265001 from LifeSpan Bioscience
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Anti-OPRK1 / Kappa Opioid Receptor Antibody (aa367-379) - LS-C139717 from LifeSpan Bioscience
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Anti-OPRK1 / Kappa Opioid Receptor Antibody (aa181-209, FITC) - LS-C265002 from LifeSpan Bioscience
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Anti-OPRK1 / Kappa Opioid Receptor Antibody (Extracellular Domain) IHC-plus⢠- LS-A228 from LifeSpan Bioscience
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