Gene Symbol | FFAR1 |
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Entrez Gene | 2864 |
Alt Symbol | FFA1R, GPCR40, GPR40 |
Species | Human |
Gene Type | protein-coding |
Description | free fatty acid receptor 1 |
Other Description | G protein-coupled receptor 40|G-protein coupled receptor 40 |
Swissprots | O14842 Q4VBL4 Q0VAS2 |
Accessions | AAB86710 ABY87912 CAD83804 O14842 BC039436 BC095536 AAH95536 BC120943 AAI20944 BC120944 AAI20945 EF611308 ABQ96386 NM_005303 NP_005294 |
Function | G-protein coupled receptor for medium and long chain saturated and unsaturated fatty acids that plays an important role in glucose homeostasis. Fatty acid binding increases glucose- stimulated insulin secretion, and may also enhance the secretion of glucagon-like peptide 1 (GLP-1). May also play a role in bone homeostasis; receptor signaling activates pathways that inhibit osteoclast differentiation (By similarity). Ligand binding leads to a conformation change that triggers signaling via G-proteins that activate phospholipase C, leading to an increase of the intracellular calcium concentration. Seems to act through a G(q) and G(i)-mediated pathway. {ECO:0000250|UniProtKB:Q76JU9, ECO:0000269|PubMed:12496284, ECO:0000269|PubMed:17699519, ECO:0000269|PubMed:24130766}. |
Subcellular Location | Cell membrane {ECO:0000269|PubMed:17699519, ECO:0000269|PubMed:25043059}; Multi-pass membrane protein {ECO:0000269|PubMed:25043059}. |
Tissue Specificity | Detected in brain and pancreas. Detected in pancreatic beta cells. {ECO:0000269|PubMed:12496284, ECO:0000269|PubMed:16289108}. |
GPR40 CRISPR/Cas9 KO Plasmid (h) - sc-401434 from Santa Cruz Biotechnology
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GPR40 HDR Plasmid (h) - sc-401434-HDR from Santa Cruz Biotechnology
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GPR40 Double Nickase Plasmid (h) - sc-401434-NIC from Santa Cruz Biotechnology
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GPR40 Double Nickase Plasmid (h2) - sc-401434-NIC-2 from Santa Cruz Biotechnology
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GPR40 CRISPR Activation Plasmid (h) - sc-401434-ACT from Santa Cruz Biotechnology
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GPR40 CRISPR Activation Plasmid (h2) - sc-401434-ACT-2 from Santa Cruz Biotechnology
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GPR40 Lentiviral Activation Particles (h) - sc-401434-LAC from Santa Cruz Biotechnology
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GPR40 Lentiviral Activation Particles (h2) - sc-401434-LAC-2 from Santa Cruz Biotechnology
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GPR40 siRNA (h) - sc-105408 from Santa Cruz Biotechnology
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GPR40 shRNA Plasmid (h) - sc-105408-SH from Santa Cruz Biotechnology
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GPR40 shRNA (h) Lentiviral Particles - sc-105408-V from Santa Cruz Biotechnology
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FFAR1/GPR40 RNAi - H00002864-R02 from Novus Biologicals
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CompoZr® Knockout ZFN Kit - CKOZFN8635 from Sigma-Aldrich
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CompoZr® Knockout ZFN Kit, ZFN plasmid only - CKOZFND8635 from Sigma-Aldrich
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CompoZr® Knockout ZFN Kit, ZFN plasmid only - CKOZFND1104 from Sigma-Aldrich
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FFAR1 siRNA (Human) - CRH1923 from Cohesion Biosciences
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FFAR1 - MBS8202573 from MyBioSource
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GPR40 CRISPR/Cas9 KO Plasmid (h2) - sc-401434-KO-2 from Santa Cruz Biotechnology
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GPR40 HDR Plasmid (h2) - sc-401434-HDR-2 from Santa Cruz Biotechnology
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shRNA set against Human FFAR1 (NM_005303.2) - SHH294229 from Creative biogene
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Human FFAR1 siRNA - orb262425 from Biorbyt
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FFAR1 shRNA Plasmid (Human) - CHH1923 from Cohesion Biosciences
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FFAR1 miRNA 3'UTR clone - MiUTR4H-TG03521 from Creative biogene
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