Gene Symbol | GCKR |
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Entrez Gene | 2646 |
Alt Symbol | FGQTL5, GKRP |
Species | Human |
Gene Type | protein-coding |
Description | glucokinase (hexokinase 4) regulator |
Other Description | glucokinase regulatory protein |
Swissprots | Q99522 Q53RY6 Q14397 B4DPQ2 A1L4C2 |
Accessions | AAP72013 AAY14850 CAA70779 CAB61828 EAX00568 Q14397 AK291846 BAF84535 AK298448 BAG60664 AK303784 BAG64742 AK309599 BC130481 AAI30482 BC130483 AAI30484 CD368544 DA011063 HQ258318 ADR83072 Z48475 CAA88367 XM_011532761 XP_011531063 XM_011532762 XP_011531064 XM_011532763 XP_011531065 NM_001486 NP_001477 |
Function | Inhibits glucokinase (GCK) by forming an inactive complex with this enzyme. The affinity of GCKR for GCK is modulated by fructose metabolites: GCKR with bound fructose 6- phosphate has increased affinity for GCK, while GCKR with bound fructose 1-phosphate has strongly decreased affinity for GCK and does not inhibit GCK activity. {ECO:0000269|PubMed:23621087, ECO:0000269|PubMed:23733961}. |
Subcellular Location | Cytoplasm {ECO:0000269|PubMed:10456334}. Nucleus {ECO:0000269|PubMed:10456334}. Note=Under low glucose concentrations, GKRP associates with GCK and the inactive complex is recruited to the hepatocyte nucleus. |
Tissue Specificity | Found in liver and pancreas. Not detected in muscle, brain, heart, thymus, intestine, uterus, adipose tissue, kidney, adrenal, lung or spleen. {ECO:0000269|PubMed:19643913, ECO:0000269|PubMed:9570959}. |
GCKR CRISPR/Cas9 KO Plasmid (h) - sc-401623 from Santa Cruz Biotechnology
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GCKR HDR Plasmid (h) - sc-401623-HDR from Santa Cruz Biotechnology
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GCKR Double Nickase Plasmid (h) - sc-401623-NIC from Santa Cruz Biotechnology
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GCKR Double Nickase Plasmid (h2) - sc-401623-NIC-2 from Santa Cruz Biotechnology
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GCKR CRISPR Activation Plasmid (h) - sc-401623-ACT from Santa Cruz Biotechnology
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GCKR CRISPR Activation Plasmid (h2) - sc-401623-ACT-2 from Santa Cruz Biotechnology
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GCKR Lentiviral Activation Particles (h) - sc-401623-LAC from Santa Cruz Biotechnology
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GCKR Lentiviral Activation Particles (h2) - sc-401623-LAC-2 from Santa Cruz Biotechnology
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GCKR siRNA (h) - sc-35460 from Santa Cruz Biotechnology
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GCKR shRNA Plasmid (h) - sc-35460-SH from Santa Cruz Biotechnology
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GCKR shRNA (h) Lentiviral Particles - sc-35460-V from Santa Cruz Biotechnology
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MISSION® esiRNA - EHU120941 from Sigma-Aldrich
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CompoZr® Knockout ZFN Kit - CKOZFN9190 from Sigma-Aldrich
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CompoZr® Knockout ZFN Kit, ZFN plasmid only - CKOZFND9190 from Sigma-Aldrich
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MISSION® 3′UTR Lenti GoClone™ - HUTR01734 from Sigma-Aldrich
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GCKR siRNA (Human) - CRH1760 from Cohesion Biosciences
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GCKR - MBS8212417 from MyBioSource
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shRNA set against Human GCKR (NM_001486.3) - SHH300034 from Creative biogene
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GCKR shRNA Plasmid (Human) - CHH1760 from Cohesion Biosciences
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GCKR miRNA 3'UTR clone - MiUTR3H-03671 from Creative biogene
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